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Chemical Structure : VU6028418
CAS No.: 2649803-05-2
Catalog No.: PC-72783Not For Human Use, Lab Use Only.
VU6028418 (VU 6028418) is a potent, highly selective, orally bioavailable M4 mAChR antagonist with IC50 of 4.1 nM (hM4).
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $348 | In stock | |
| 10 mg | $548 | In stock | |
| 25 mg | Get quote | ||
| 100 mg | Get quote |
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VU6028418 (VU 6028418) is a potent, highly selective, orally bioavailable M4 mAChR antagonist with IC50 of 4.1 nM (hM4).
| M.Wt | 432.491 | |
| Formula | C23H27F3N4O | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
rel-(3aR,6aS)-Octahydro-2-[(tetrahydro-2H-pyran-4-yl)methyl]-N-[6-(2,3,5-trifluorophenyl)-3-pyridazinyl]cyclopenta[c]pyrrol-5-amine |
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1. Matthew Spock, et al. ACS Med Chem Lett. 2021 Aug 2;12(8):1342-1349.
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