Welcome to ProbeChem!Global Supplier of Chemical Probes, Inhibitors & Agonists.
    English |     Chinese

Product Inquiry: sales@probechem.com
Order/PO receiving: order@probechem.com

You are here:Home-Chemical Inhibitors & Agonists-GPCR-mAChR-VU6028418
VU6028418

Chemical Structure : VU6028418

CAS No.: 2649803-05-2

Add to Favorites

VU6028418 (VU 6028418)

Catalog No.: PC-72783Not For Human Use, Lab Use Only.

VU6028418 (VU 6028418) is a potent, highly selective, orally bioavailable M4 mAChR antagonist with IC50 of 4.1 nM (hM4).

Packing Price Stock Quantity
5 mg $348 In stock
10 mg $548 In stock
25 mg Get quote
100 mg Get quote
Get Quotation Now
* Please select Quantity before adding items.
 or Bulk Inquiry

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

VU6028418 (VU 6028418) is a potent, highly selective, orally bioavailable M4 mAChR antagonist with IC50 of 4.1 nM (hM4).

Physicochemical Properties

M.Wt 432.491
Formula C23H27F3N4O
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

rel-(3aR,6aS)-Octahydro-2-[(tetrahydro-2H-pyran-4-yl)methyl]-N-[6-(2,3,5-trifluorophenyl)-3-pyridazinyl]cyclopenta[c]pyrrol-5-amine

References

1. Matthew Spock, et al. ACS Med Chem Lett. 2021 Aug 2;12(8):1342-1349.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: