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Chemical Structure : VU6036864
Catalog No.: PC-22893Not For Human Use, Lab Use Only.
VU6036864 is a highly potent, selective antagonist of muscarinic acetylcholine receptor mAChR subtype 5 (M5) with IC50 of 25 nM (hM5), >500 fold selectivity against M1-4 receptors.
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VU6036864 is a highly potent, selective antagonist of muscarinic acetylcholine receptor mAChR subtype 5 (M5) with IC50 of 25 nM (hM5), >500 fold selectivity against M1-4 receptors.
VU6036864 exhibited good potency, subtype selectivity, and oral DMPK properties.
| M.Wt | 385.86 | |
| Formula | C15H12D4ClN5O3S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Jinming Li, et al. J Med Chem. 2024 Aug 6. doi: 10.1021/acs.jmedchem.4c01193.
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