VU6069863 | M1 PAM | Probechem Biochemicals

Chemical Structure : VU6069863

Catalog No.: PC-28266Not For Human Use, Lab Use Only.

VU6069863 is a potent, selective M1 positive allosteric modulator (PAM) with EC50 of 226 nM and 140 nM for hM1 and rM1, shows minimal M1 agonism.

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Biological Activity

VU6069863 is a potent, selective M1 positive allosteric modulator (PAM) with EC50 of 226 nM and 140 nM for hM1 and rM1, shows minimal M1 agonism.

M.Wt	348.40
Formula	C21H20N2O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	8,9-dimethyl-7-(4-(oxazol-4-yl)benzyl)-3,4-dihydrobenzo[f][1,4]oxazepin-5(2H)-one

1. Changho Han, et al. ACS Med Chem Lett. 2026 Aug 21;17(9):2085-2094.