VUF15000 | Probechem Biochemicals

Chemical Structure : VUF15000

VUF15000 (VUF-15000;VUF 15000)

Catalog No.: PC-36072Not For Human Use, Lab Use Only.

VUF15000 (VUF-15000) is the first photoswitchable GPCR Histamine H3 receptor agonist (pKi=8.42), displays >300-fold selective for hH3R over hH1R and hH2R.

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Biological Activity

VUF15000 (VUF-15000) is the first photoswitchable GPCR Histamine H3 receptor agonist (pKi=8.42), displays >300-fold selective for hH3R over hH1R and hH2R.
VUF15000 induces Gi activation with pEC50 of 7.60.
VUF15000 is a new chemical biology tool for spatiotemporal control of GPCR activation.

Physicochemical Properties

M.Wt	262.316
Formula	C16H14N4
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Trans-4-(3-(phenyldiazenyl)benzyl)-1H-imidazole

References

1. Hauwert NJ, et al. Angew Chem Int Ed Engl. 2019 Feb 8. doi: 10.1002/anie.201813110.

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VUF15000 (VUF-15000;VUF 15000)

Biological Activity

Physicochemical Properties

References

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