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Chemical Structure : VUF15000
Catalog No.: PC-36072Not For Human Use, Lab Use Only.
VUF15000 (VUF-15000) is the first photoswitchable GPCR Histamine H3 receptor agonist (pKi=8.42), displays >300-fold selective for hH3R over hH1R and hH2R.
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VUF15000 (VUF-15000) is the first photoswitchable GPCR Histamine H3 receptor agonist (pKi=8.42), displays >300-fold selective for hH3R over hH1R and hH2R.
VUF15000 induces Gi activation with pEC50 of 7.60.
VUF15000 is a new chemical biology tool for spatiotemporal control of GPCR activation.
| M.Wt | 262.316 | |
| Formula | C16H14N4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Hauwert NJ, et al. Angew Chem Int Ed Engl. 2019 Feb 8. doi: 10.1002/anie.201813110.
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