Varenicline | α4β2 nAChR agonist | Probechem Biochemicals

Chemical Structure : Varenicline

CAS No.: 249296-44-4

Varenicline (CP 526555)

Catalog No.: PC-26759Not For Human Use, Lab Use Only.

Varenicline (CP 526555) is a potent, orally active partial agonist of α4β2 nicotinic acetylcholine receptor (α4β2 nAChR) with IC50 of 250 nM, is also a partial agonist of α6β2 nAChR and a full agonist of α7β2 nAChR.

Packing	Price	Stock
10 mg	$78	In stock
25 mg	$128	In stock
50 mg	$198	In stock
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Biological Activity

Physicochemical Properties

M.Wt	211.27
Formula	C13H13N3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	7,8,9,10-Tetrahydro-6H-6,10-methanoazepino[4,5-g]quinoxaline

References

1. Koegelenberg CF, et al. JAMA. 2014 Jul;312(2):155-61.

2. Koga M, et al. Toxicology. 2017;390:1-9.

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Varenicline (CP 526555)

Biological Activity

Physicochemical Properties

References

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