Chemical Structure : Varenicline Tartrate
CAS No.: 375815-87-5
Catalog No.: PC-26760Not For Human Use, Lab Use Only.
Varenicline Tartrate (CP 526555) is a potent, orally active partial agonist of α4β2 nicotinic acetylcholine receptor (α4β2 nAChR) with IC50 of 250 nM, is also a partial agonist of α6β2 nAChR and a full agonist of α7β2 nAChR.
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|---|---|---|---|
| 25 mg | $78 | In stock | |
| 50 mg | $128 | In stock | |
| 100 mg | $198 | In stock | |
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Varenicline Tartrate (CP 526555) is a potent, orally active partial agonist of α4β2 nicotinic acetylcholine receptor (α4β2 nAChR) with IC50 of 250 nM, is also a partial agonist of α6β2 nAChR and a full agonist of α7β2 nAChR.
| M.Wt | 361.35 | |
| Formula | C17H19N3O6 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
7,8,9,10-Tetrahydro-6H-6,10-methanoazepino[4,5-g]quinoxaline tartrate |
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1. Koegelenberg CF, et al. JAMA. 2014 Jul;312(2):155-61.
2. Koga M, et al. Toxicology. 2017;390:1-9.

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