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You are here:Home-Chemical Inhibitors & Agonists-GPCR-Mas-related G protein-coupled receptor (MRGPR)-ZINC-3573 racemate
ZINC-3573 racemate

Chemical Structure : ZINC-3573 racemate

CAS No.: 1378183-16-4

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ZINC-3573 racemate (ZINC3573 racemate)

Catalog No.: PC-62228Not For Human Use, Lab Use Only.

ZINC-3573 racemate is a potent, selective agonist of the atypical opioid receptor MRGPRX2 (EC50=3 uM), showing little activity against 315 other GPCRs and 97 representative kinases.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    ZINC-3573 racemate is a potent, selective agonist of the atypical opioid receptor MRGPRX2 (EC50=3 uM), showing little activity against 315 other GPCRs and 97 representative kinases.
    ZINC-3573 activates endogenous MRGPRX2 in a human mast cell line, inducing degranulation and calcium release.

    Physicochemical Properties

    M.Wt 307.401
    Formula C18H21N5
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    Dimethyl-[1-(5-phenyl-pyrazolo[1,5-a]pyrimidin-7-yl)-pyrrolidin-3-yl]-amine

    References

    1. Lansu K, et al. Nat Chem Biol. 2017 May;13(5):529-536.

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