Zamicastat | Dopamine beta-hydroxylase inhibitor

Chemical Structure : Zamicastat

CAS No.: 1080028-80-3

Catalog No.: PC-22596Not For Human Use, Lab Use Only.

Zamicastat (BIA 5-1058) is a potent, selective dopamine β-hydroxylase (DβH) inhibitor, decreases noradrenaline and increases dopamine levels.

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Biological Activity

Zamicastat (BIA 5-1058) is a potent, selective dopamine β-hydroxylase (DβH) inhibitor, decreases noradrenaline and increases dopamine levels.

M.Wt	401.48
Formula	C21H21F2N3OS
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1-[(3R)-6,8-Difluoro-3,4-dihydro-2H-1-benzopyran-3-yl]-1,3-dihydro-5-[2-[(phenylmethyl)amino]ethyl]-2H-imidazole-2-thione

1. Igreja B, et al. Eur J Pharmacol. 2019 Jan 5;842:125-132.

2. Bicker J, et al. Eur J Pharm Sci. 2018 May 30;117:35-40.