Chemical Structure : Zatebradine
CAS No.: 85175-67-3
Catalog No.: PC-43527Not For Human Use, Lab Use Only.
Zatebradine (UL-FS49) is a potent blocker (antagonist) of hyperpolarization-activated cyclic nucleotide-gated (HCN) channel, a specific bradycardic agent.
Packing | Price | Stock | Quantity |
---|---|---|---|
5 mg | $58 | In stock | |
10 mg | $88 | In stock | |
25 mg | $148 | In stock | |
50 mg | $258 | In stock | |
100 mg | Get quote |
Bulk size, bulk discount!
Welcome credit card payment!
E-mail: sales@probechem.com
Tech Support: tech@probechem.com
Zatebradine (UL-FS49) is a potent blocker (antagonist) of hyperpolarization-activated cyclic nucleotide-gated (HCN) channel, a specific bradycardic agent.
Zatebradine (UL-FS49) blocks cardiac pacemaker current (If), decreases the rate of spontaneously beating guinea-pig atria with EC50 of 0.030 ug/mL.
M.Wt | 456.5744 | |
Formula | C26H36N2O5 | |
Appearance | Solid | |
Storage |
|
|
Solubility |
10 mM in DMSO |
|
Chemical Name/SMILES |
2H-3-Benzazepin-2-one, 3-[3-[[2-(3,4-dimethoxyphenyl)ethyl]methylamino]propyl]-1,3,4,5-tetrahydro-7,8-dimethoxy- |
1. Van Bogaert PP, et al. Eur J Pharmacol. 2003 Oct 8;478(2-3):161-71.
2. McGovern AE, et al. Br J Pharmacol. 2014 Aug;171(15):3633-50.
3. Gill CH, et al. Br J Pharmacol. 2004 Oct;143(3):411-21.
Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright