Chemical Structure : Zibotentan
CAS No.:
186497-07-4
Zibotentan
(ZD4054, ZD-4054)
Catalog No. : PC-42282Not For Human Use, Lab Use Only.
Zibotentan (ZD4054) is an orally active, specific Endothelin A receptor (ETA) inhibitor with Ki of 13 nM, shows anticancer effects.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4228201
Biological Activity
Zibotentan (ZD4054) is an orally active, specific Endothelin A receptor (ETA) inhibitor with Ki of 13 nM, shows anticancer effects.
Physicochemical Properties
M.Wt
424.4331
Formula
C19H16N6O4S
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
3-Pyridinesulfonamide, N-(3-methoxy-5-methyl-2-pyrazinyl)-2-[4-(1,3,4-oxadiazol-2-yl)phenyl]-
References
1. Morris CD, et al. Br J Cancer.
2. Bradbury RH, et al. J Med Chem.
3. Carducci MA, et al. Clin Cancer Res.
4. Rosanò L, et al. Mol Cancer Ther.
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