Chemical Structure : (-)-GSK598809
CAS No.:
863680-46-0
(-)-GSK598809
(GSK598809)
Catalog No. : PC-49576Not For Human Use, Lab Use Only.
GSK598809 (GSK-598809) is a potent, selective dopamine D(3) receptor antagonist with Ki value of 6.2 nM, >100-fold selectivity over D2 receptor.
Packing Price Stock Quantity 5 mg $148 In stock 0 1 2 3 4 5 10 mg $218 In stock 0 1 2 3 4 5 25 mg $378 In stock 0 1 2 3 4 5 50 mg $588 In stock 0 1 2 3 4 5 100 mg Get quote 0 1 2 3 4 5
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4957601
Biological Activity
GSK598809 (GSK-598809) is a potent, selective dopamine D(3) receptor antagonist with Ki value of 6.2 nM, >100-fold selectivity over D2 receptor.
Physicochemical Properties
M.Wt
481.51
Formula
C22H23F4N5OS
Appearance
Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
5-(5-((3-((1S,5R)-1-(2-fluoro-4-(trifluoromethyl)phenyl)-3-azabicyclo[3.1.0]hexan-3-yl)propyl)thio)-4-methyl-4H-1,2,4-triazol-3-yl)-4-methyloxazole
References
1. Searle G, et al. Biol Psychiatry. 2010 Aug 15;68(4):392-9.
2. Appel NM, et al. J Pharmacol Exp Ther. 2015 Sep;354(3):484-92.
3. Mugnaini M, et al. Neuropsychopharmacology. 2013 Jan;38(2):302-12.
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