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Chemical Structure : 5-BDBD
CAS No.: 768404-03-1
Catalog No.: PC-72721Not For Human Use, Lab Use Only.
5-BDBD is a potent and selective P2X4 receptor (P2X4R) antagonist, inhibits P2X4-mediated currents in CHO cells with IC50 of 0.5 uM.
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|---|---|---|---|
| 10 mg | $158 | In stock | |
| 25 mg | $258 | In stock | |
| 50 mg | $398 | In stock | |
| 100 mg | Get quote |
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5-BDBD is a potent and selective P2X4 receptor (P2X4R) antagonist, inhibits P2X4-mediated currents in CHO cells with IC50 of 0.5 uM.
5-BDBD displays no significant antagonist effects at other P2X receptors.
5-BDBD reduces long-term potentiation (LTP) in rat hippocampal slices.
| M.Wt | 355.191 | |
| Formula | C17H11BrN2O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
5-(3-bromophenyl)-1,3-dihydro-2H-benzofuro[3,2-e]-1,4-diazepin-2-one |
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1. Wu T, et al. Am J Physiol Heart Circ Physiol. 2011 Jul;301(1):H69-78.
2. Balázs B, et al. Cell Physiol Biochem. 2013;32(1):11-24.
3. Barr TP, et al. Pain. 2014 Jun;155(6):1091-1101.
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