5-BDBD

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Chemical Structure : 5-BDBD

CAS No.: 768404-03-1

Catalog No.: PC-72721Not For Human Use, Lab Use Only.

5-BDBD is a potent and selective P2X4 receptor (P2X4R) antagonist, inhibits P2X4-mediated currents in CHO cells with IC50 of 0.5 uM.

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10 mg	$158	In stock
25 mg	$258	In stock
50 mg	$398	In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

5-BDBD is a potent and selective P2X4 receptor (P2X4R) antagonist, inhibits P2X4-mediated currents in CHO cells with IC50 of 0.5 uM.
5-BDBD displays no significant antagonist effects at other P2X receptors.
5-BDBD reduces long-term potentiation (LTP) in rat hippocampal slices.

Physicochemical Properties

M.Wt	355.191
Formula	C17H11BrN2O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	5-(3-bromophenyl)-1,3-dihydro-2H-benzofuro[3,2-e]-1,4-diazepin-2-one

References

1. Wu T, et al. Am J Physiol Heart Circ Physiol. 2011 Jul;301(1):H69-78.

2. Balázs B, et al. Cell Physiol Biochem. 2013;32(1):11-24.

3. Barr TP, et al. Pain. 2014 Jun;155(6):1091-1101.

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5-BDBD

Biological Activity

Physicochemical Properties

References

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