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A-68930 hydrochloride

Chemical Structure : A-68930 hydrochloride

CAS No.: 130465-39-3

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A-68930 hydrochloride (A68930)

Catalog No.: PC-63113Not For Human Use, Lab Use Only.

A-68930 is a potent, specific, orally bioavailable agonist of the D1 dopamine receptor (D1DR) with EC50 of 2.5 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    A-68930 is a potent, specific, orally bioavailable agonist of the D1 dopamine receptor (D1DR) with EC50 of 2.5 nM.
    A-68930 shows a much weaker agonist (EC50=3,920 nM) at the D2 dopamine receptor.
    A-68930 demonstrates antidepressant and anorectic effects in animal models without stimulant effects.

    Physicochemical Properties

    M.Wt 307.77
    Formula C16H17NO3 · HCl
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    1H-2-Benzopyran-5,6-diol, 1-(aminomethyl)-3,4-dihydro-3-phenyl-, hydrochloride, (1R,3S)-rel- (9CI)

    References

    1. Kebabian JW, et al. Am J Hypertens. 1990 Jun;3(6 Pt 2):40S-42S.

    2. Trampus M, et al. Eur J Pharmacol. 1993 Apr 22;235(1):83-7.

    3. AI-Naser HA, et al. Behav Pharmacol. 1994 Apr;5(2):210-218.

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