Chemical Structure : A-804598
CAS No.:
1125758-85-1
A-804598
(A 804598, A804598)
Catalog No. : PC-42169Not For Human Use, Lab Use Only.
A-804598 is a potent, selective and competitive P2X7 receptor antagonist with IC50 of 10, 9 , and 11 nM for rat, mouse, and human P2X7, respectively.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4216901
Biological Activity
A-804598 is a potent, selective and competitive P2X7 receptor antagonist with IC50 of 10, 9 , and 11 nM for rat, mouse, and human P2X7, respectively.
Physicochemical Properties
M.Wt
315.3718
Formula
C19H17N5
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
DMSO: ≥ 32 mg/mL
Chemical Name/SMILES
Guanidine, N-cyano-N''-[(1S)-1-phenylethyl]-N'-5-quinolinyl-
References
1. Donnelly-Roberts DL, et al. Neuropharmacology.
2. Catanzaro JM, et al. Behav Pharmacol.
3. Ziff J, et al. ACS Chem Neurosci.
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