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Chemical Structure : ACT-539313
Catalog No.: PC-21251Not For Human Use, Lab Use Only.
Nivasorexant (ACT-539313) is a potent, selective and brain-penetrating orexin receptor type 1 receptor (OX1R) antagonist with Kb of 0.69 nM (human OX1R), 60-fold selective over OX2R.
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Nivasorexant (ACT-539313) is a potent, selective and brain-penetrating orexin receptor type 1 receptor (OX1R) antagonist with Kb of 0.69 nM (human OX1R), 60-fold selective over OX2R.
Nivasorexant (ACT-539313) shows potential in the treatment of humans with binge-eating disorder.
| M.Wt | 429.48 | |
| Formula | C23H23N7O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Berger B, et al. J Clin Pharmacol. 2020 Jul;60(7):931-941.
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