AKR1C3 inhibitor 1

Chemical Structure : AKR1C3 inhibitor 1

Catalog No.: PC-22254Not For Human Use, Lab Use Only.

AKR1C3 inhibitor 1 is a potent, selective aldo-keto reductase 1C3 (AKR1C3) inhibitor with IC50 of 110 nM, 127-fold selective over AKR1C2.

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Biological Activity

AKR1C3 inhibitor 1 is a potent, selective aldo-keto reductase 1C3 (AKR1C3) inhibitor with IC50 of 43 nM, >2300-fold selective over AKR1C2.

M.Wt	371.44
Formula	C24H21NO3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(E)-3-(5-((4-methylbenzyl)carbamoyl)-[1,1'-biphenyl]-3-yl)acrylic acid

1. Carmona AV, et al. Commun Chem. 2024 Apr 29;7(1):95.