Welcome to ProbeChem!Global Supplier of Chemical Probes, Inhibitors & Agonists.

You are here:Home-Chemical Inhibitors & Agonists-GPCR-Cannabinoid Receptor-AM10257
AM10257

Chemical Structure : AM10257

CAS No.: 2316841-32-2

AM10257 (AM-10257)

Catalog No.: PC-22167Not For Human Use, Lab Use Only.

AM10257 is a potent, selective cannabinoid receptor 2 (CB2) antagonist with IC50 of 47 nM.

Packing Price Stock Quantity
25 mg Get quote
50 mg Get quote
100 mg Get quote
250 mg Get quote

Bulk size, bulk discount!

Welcome credit card payment!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC)

Biological Activity

AM10257 is a potent, selective cannabinoid receptor 2 (CB2) antagonist with IC50 of 47 nM.

Physicochemical Properties

M.Wt 421.59
Formula C26H35N3O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

N-(adamantan-1-yl)-1-(5-hydroxypentyl)-4-methyl-5-phenyl-1H-pyrazole-3-carboxamide

References

1. Hu T, et al. J Med Chem. 2021 Sep 23;64(18):13752-13765.

2. Li X, et al. Cell. 2019 Jan 24;176(3):459-467.e13.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: