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AM630

Chemical Structure : AM630

CAS No.: 164178-33-0

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AM630 (AM-630, 6-Iodopravodoline)

Catalog No.: PC-60760Not For Human Use, Lab Use Only.

AM630 (6-Iodopravodoline) is a potent and selective inverse agonist for the cannabinoid receptor CB2 with Ki of 32.1 nM, 165-fold selectivity over CB1.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

AM630 (6-Iodopravodoline) is a potent and selective inverse agonist for the cannabinoid receptor CB2 with Ki of 32.1 nM, 165-fold selectivity over CB1.
AM630 inhibits forskolin-stimulated cyclic AMP production in CB1-transfected cells (22.6% at 1 uM and 45.9% at 10 uM).

Physicochemical Properties

M.Wt 504.4
Formula C23H25IN2O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

[6-iodo-2-methyl-1-[2-(4-morpholinyl)ethyl]-1H-indol-3-yl](4-methoxyphenyl)-methanone

References

1. Ross RA, et al. Br J Pharmacol. 1999 Feb;126(3):665-72.

2. Malan TP Jr, et al. Pain. 2001 Sep;93(3):239-45.

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