AMG2504 | TRPA1 inhibitor | Probechem Biochemicals

Chemical Structure : AMG2504

AMG2504 (AMG 2504)

Catalog No.: PC-49701Not For Human Use, Lab Use Only.

AMG2504 (AMG 2504) is a selective small molecule TRPA1 inhibitor, inhibits AITC-induced increase in intracellular calcium mediated by TRPA1 in CHO cells with IC50 of 35 nM.

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Biological Activity

AMG2504 (AMG 2504) is a selective small molecule TRPA1 inhibitor, inhibits AITC-induced increase in intracellular calcium mediated by TRPA1 in CHO cells with IC50 of 35 nM.
AMG2504 displays no activity against hTRPV1, hTRPM8, hTRPV3 and hTRPV4 at 5 uM.
AMG2504 marginally inhibited rat TRPA1 activation by AITC.

Physicochemical Properties

M.Wt	440.12
Formula	C15H10Cl4N2O3S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	4-nitro-N-(2,2,2-trichloro-1-((4-chlorophenyl)thio)ethyl)benzamide

References

1. Lana Klionsky, et al. Mol Pain. 2007 Dec 17;3:39. doi: 10.1186/1744-8069-3-39.

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AMG2504 (AMG 2504)

Biological Activity

Physicochemical Properties

References

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