Chemical Structure : AMG517
CAS No.:
659730-32-2
AMG517
(AMG 517, AMG-517)
Catalog No. : PC-42689Not For Human Use, Lab Use Only.
AMG517 is a potent and selective vanilloid receptor TRPV1 antagonist with IC50 of 0.76 nM for hTRPV
Packing Price Stock Quantity 5 mg (Free Sample) $28 In stock 0 1 2 3 4 5 10 mg $78 In stock 0 1 2 3 4 5 25 mg $138 In stock 0 1 2 3 4 5 50 mg $238 In stock 0 1 2 3 4 5 100 mg Get quote 0 1 2 3 4 5
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4268901
Biological Activity
AMG517 is a potent and selective vanilloid receptor TRPV1 antagonist with IC50 of 0.76 nM for hTRPV1.
Physicochemical Properties
M.Wt
430.403
Formula
C20H13F3N4O2S
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
DMSO: 12.91 mg/mL (Need ultrasonic)
Chemical Name/SMILES
Acetamide, N-[4-[[6-[4-(trifluoromethyl)phenyl]-4-pyrimidinyl]oxy]-2-benzothiazolyl]-
References
1. Doherty EM, et al. J Med Chem
2. Gavva NR, et al. J Pharmacol Exp Ther.
3. Gavva NR, et al. Pain
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