ARN25068 | GSK-3β/FYN/DYRK1A inhibitor

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Chemical Structure : ARN25068

CAS No.: 2649882-80-2

ARN25068 (ARN-25068)

Catalog No.: PC-38653Not For Human Use, Lab Use Only.

ARN25068 is a highly potent, triple GSK-3β/FYN/DYRK1A inhibitor with IC50 of 4.17 and 2.17 μM for GSK-3β and FYN, reduces the extent of tau phosphorylation in Tau0N4R-TM-tGFP U2OS cell line.

Packing	Price	Stock
5 mg	$198	In stock
10 mg	$298	In stock
25 mg	$498	In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

ARN25068 is a highly potent, triple GSK-3β/FYN/DYRK1A inhibitor with IC50 of 4.17 and 2.17 μM for GSK-3β and FYN, reduces the extent of tau phosphorylation in Tau0N4R-TM-tGFP U2OS cell line.

Physicochemical Properties

M.Wt	362.455
Formula	C19H18N6S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	N2-benzyl-N4-(3-cyclopropyl-1H-pyrazol-5-yl)thieno[3,2-d]pyrimidine-2,4-diamine

References

1. Stefania Demuro, et al. Eur J Med Chem. 2022 Feb 5;229:114054.

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ARN25068 (ARN-25068)

Biological Activity

Physicochemical Properties

References

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