ARUK2001607 | PI5P4Kγ inhibitor | Probechem Biochemicals

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Chemical Structure : ARUK2001607

ARUK2001607 (ARUK 2001607)

Catalog No.: PC-49589Not For Human Use, Lab Use Only.

ARUK2001607 is a potent, selective and brain penetrant PI5P4Kγ inhibitor with binding KD of 7.1 nM, pIC50 of 7.1 (PI5P4Kγ+).

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

ARUK2001607 is a potent, selective and brain penetrant PI5P4Kγ inhibitor with binding KD of 7.1 nM, pIC50 of 7.1 (PI5P4Kγ+).
ARUK2001607 showed excellent selectivity data against >150 kinases and a Cerep safety panel, also showed good potencies at PI5P4Kγ (WT and γ+), were selective vs PI5P4Kα and β.

Physicochemical Properties

M.Wt	319.40
Formula	C14H13N3O2S2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	6-Methyl-N-(4-(methylsulfonyl)phenyl)thieno[2,3-d]pyrimidin-4-amine

References

1. Timothy P C Rooney, et al. J Med Chem. 2022 Dec 14. doi: 10.1021/acs.jmedchem.2c01693.

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ARUK2001607 (ARUK 2001607)

Biological Activity

Physicochemical Properties

References

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