Chemical Structure : AZD5153
CAS No.:
1869912-39-9
AZD5153
(AZD-5153)
Catalog No. : PC-62986Not For Human Use, Lab Use Only.
AZD5153 is a potent, selective, bivalent and orally available BET/BRD4 bromodomain with IC50 of 5 nM.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-6298601
Biological Activity
AZD5153 is a potent, selective, bivalent and orally available BET/BRD4 bromodomain with IC50 of 5 nM.
Physicochemical Properties
M.Wt
479.585
Formula
C25H33N7O3
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
(R)-4-(2-(4-(1-(3-methoxy-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperidin-4-yl)phenoxy)ethyl)-1,3-dimethylpiperazin-2-one
References
1. Bradbury RH, et al. J Med Chem.
2. Rhyasen GW, et al. Mol Cancer Ther.
3. Collins TA, et al. CPT Pharmacometrics Syst Pharmacol.
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