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Cat. No. Product Name CAS No. Information
PC-38071

GSK778

2451862-42-1 GSK778 is a potent and selective inhibitor of bromodomain (BRD) BD1 with IC50 of 75 nM (BRD2-BD1), 41 nM (BRD3-BD1), 41 nM (BRD4 BD1), and 143 nM (BRDT BD1), respectively.
PC-38064

ODM-207

1801503-93-4 ODM-207 (ODM207) is a highly potent, selective and orally active pan-BET inhibitor with potent and broad antiproliferative effects.
PC-35848

TP-238

2415263-04-4 TP-238 (TP238) is a CECR2/BPTF bromodomains chemical probe with IC50 of 30 nM against CECR2 and 350 nM against BPTF in an alphascreen assay, KD of 10 nM for CECR2 and 120nM for BPTF in ITC assays.
PC-35172

ABBV-744

2138861-99-9 ABBV-744 (ABBV744) is a potent, BDII-selective BET bromodomain inhibitor, ABBV-744 is a potent, selective inhibitor of the AR transcription activity.
PC-35097

ZL0454

2229042-77-5 ZL0454 is a potent, highly selective small-molecule BRD4 inhibitor with IC50 of 49 and 32 nM for BRD4-BD1 and BRD4-BD2, respectively.
PC-35096

ZL0420

2229039-45-4 ZL0420 is a potent, highly selective BRD4 inhibitor with IC50 of 27 and 32 nM for BRD4-BD1 and BRD4-BD2, respectively.
PC-63272

INCB057643

1820889-23-3 INCB057643 is a novel potent, selective, orally bioavailable BET inhibitor.

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