Bromodomain compound (inhibitors, agonists)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-21072	IV-255 BRG1 selective inhibitor	IV-255 is a next-generation selective inhibitor of BRG1 bromodomain, inhibits SWI/SNF complex and enhances DNA damage and cell death in glioblastoma.
PC-20948	DDO-8926 BET inhibitor	DDO-8926 is a potent selective inhibitor of bromodomain and extra-terminal (BET) proteins with Ki values of 15 nM (BRD4 BD1) and 9.5 nM (BRD4 BD2).
PC-20838	BBC1115 BET inhibitor	BBC1115 is a novel chemotype inhibitor of bromodomain and extra-terminal motif (BET) proteins, displays broad binding across BDs of BET proteins.
PC-20573	OTX-015 BET bromodomain inhibitor	Birabresib (OTX-015) is a potent, competitive inhibitor of BET bromodomain BRD2, BRD3, and BRD4 with EC50 of 10-19 nM, inhibits binding of BRD2, BRD3, and BRD4 to acetylated histone H4 (AcH4) with IC50 of 92-112 nM.
PC-72758	BPTF inhibitor BZ1 BPTF inhibitor	BPTF inhibitor BZ1 is a potent, selective, cell-active inhibitor of bromodomain PHD finger transcription factor (BPTF) with Kd of 6.3 nM, >350-fold selectivity over BET bromodomains.
PC-35016	IBET151-Az	IBET151-Az is a IBET151 derivative for PROTAC synthesis..
PC-43339	(R)-(-)-JQ1 Enantiomer	(R)-(-)-JQ1 Enantiomer is the stereoisomer of (+)-JQ1, (+)-JQ-1 is a potent, specific BET bromodomain BRD4 inhibitor, but (-)-JQ1 has no activity..

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