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Cat. No. Product Name Information
PC-22484

Y08207

CBP/p300 inhibitor

Y08207 is a potent, selective CBP/p300 bromodomain inhibitor with IC50 of 26.37 nM (CBP bromodomain) in HTRF assays.
PC-22483

Y08262

CBP/p300 inhibitor

Y08207 is a potent, selective CBP/p300 bromodomain inhibitor with IC50 of 73.1 nM (CBP bromodomain) in HTRF assays.
PC-22287

CDD-1302

BRDT BD2 inhibitor

CDD-1302 (CDD1302) is a potent, selective second bromodomain (BD2) of BRDT and BRD4 inhibitor with IC50 of 8 and 12 nM, >1,000-fold and 300-fold selectivity over BRDT-BD1 and BRD4-BD1.
PC-22217

Rac EBET-590

BET inhibitor

Rac EBET-590 (EBET-590 Racemate) is a small molecule BET inhibitor.
PC-22216

EBET-590

BET inhibitor

EBET-590 (ER-001251206-000) is a small molecule BET inhibitor.
PC-22204

SDU-071

BRD4-p53 inhibitor

SDU-071 is a potent small molecule BRD4-p53 PPI inhibitor with IC50 of 2.7 uM, reduces the expression of BRD4-regulated genes, such as c-Myc and Mucin 5AC, and induces cell cycle arrest and apoptosis.
PC-22158

BBC0403

BRD2 inhibitor

BBC0403 (BBC-0403) is a specific BRD2 inhibitor with binding Kd of 41.4 uM and 7.6 uM for BRD2 (BD1) and BRD2 (BD2), inhibits the NF-κB and MAPK signalling pathways and the progression of osteoarthritis pathogenesis.
PC-21995

ZM145

pBRD4 inhibitor

ZM145 (pNPS145) is a small molecule inhibitor of phospho-BRD4 (pBRD4) with IC50 of 2.5 uM, binds to phospho-NPS (pNPS) and disrupts HPV E2-BRD4 interaction, effectively inhibits HPV ecDNA replication.
PC-21994

pNPS90

pBRD4 inhibitor

pNPS90 is a small molecule inhibitor of phospho-BRD4 (pBRD4) with IC50 of 1.5 uM, binds to phospho-NPS (pNPS) and disrupts HPV E2-BRD4 interaction, effectively inhibits HPV ecDNA replication.
PC-21993

pNPS14

pBRD4 inhibitor

pNPS14 is a small molecule inhibitor of phospho-BRD4 (pBRD4) with IC50 of 3.39 uM, binds to phospho-NPS (pNPS) and disrupts HPV E2-BRD4 interaction, effectively inhibits HPV ecDNA replication.
PC-21985

CBP bromodomain inhibitor 29

CBP bromodomain inhibitor

CBP-IN-29 is a potent, selective CBP bromodomain inhibitor with IC50 of 2.2 nM, displays exquisite selectivity over BRD4(1) (IC50=23 uM) and the broader bromodomain family.
PC-21984

CBP bromodomain inhibitor 27

CBP bromodomain inhibitor

CBP-IN-27 is a potent, selective CBP bromodomain inhibitor with IC50 of 3.6 nM, displays exquisite selectivity over BRD4(1) (IC50=11 uM) and the broader bromodomain family.

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