Y06014 | BET inhibitor | Probechem Biochemicals

Chemical Structure : Y06014

Y06014 (Y 06014)

Catalog No.: PC-22992Not For Human Use, Lab Use Only.

Y06014 is a selective BRD4(1) inhibitor with IC50 of 4.87 uM.

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Biological Activity

Y06014 is a selective BRD4(1) inhibitor with IC50 of 4.87 uM.
Y06014 shows exhibits excellent selectivity for the BET subfamily over other non-BET families.
Y06014 shows cell viability inhibition IC50 values of 1.93, 2.07, and 2.28 μM in the C4–2B, LNCaP, and 22Rv1 cell lines, respectively.
Y06014 inhibits prostate cancer cell growth and AR-regulated gene expression.

Physicochemical Properties

M.Wt	292.34
Formula	C18H16N2O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	6-(3,5-Dimethylisoxazol-4-yl)-1-ethylbenzo[cd]indol-2(1H)-one

References

1. Tian-Bang Wu, et al. Acta Pharmacol Sin. 2021 Dec;42(12):2120-2131.

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Y06014 (Y 06014)

Biological Activity

Physicochemical Properties

References

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