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Cat. No. Product Name Information
PC-60104

HJB97

BET inhibitor

HJB-97 (HJB97) is a potent BET bromodomian inhibitor with IC50 of 3-7 nM for BRD2/3/4 BD1 and BD2.
PC-70031

PF-CBP1

CBP/p300 inhibitor

PF-CBP1 is a potent, highly selective CBP/p300 bromodomains inhibitor with IC50 of 125 nM and 363 nM, respectively.
PC-70026

CPI-268456

BRD4 inhibitor

CPI-268456 is a small molecule ligand of bromodomain-containing protein 4 (BRD4), binds to BRD4 with IC50 of 0.5 uM in cell-free assays.
PC-60022

BAY-850

ATAD2 inhibitor

BAY-850 (BAY 850, BAY850) is a potent, isoform selective, cellularly active ATAD2 bromodomain inhibitor with binding IC50 of 166 nM in TR-FRET assay.
PC-45582

I-BRD9

BRD9 inhibitor

I-BRD9 is the first selective cellular chemical probe inhibitor for BRD9 with pIC50 of 7.3.
PC-45508

GSK-5959

BRPF1 inhibitor

GSK-5959 (GSK5959) is the first potent, selective inhibitor of the BRPF1 bromodomain with pIC50 of 7.1.
PC-45994

JQ-1 carboxylic acid

BET inhibitor

JQ-1 carboxylic acid is an inhibitor of bromodomain and extra terminal domain (BET) family proteins with Kd of 128, 59.5, 49.0, and 190 nM for JQ1 binding to bromodomains of BRD2, BRD3, BRD4, and BRDT, respectively, blocking their interaction with acetylated histones.
PC-42110

BI-9564

BRD9 inhibitor

BI-9564 (BI9564) is a potent, selective, cell-permeable and noncytotoxic BRD9 bromodomain inhibitor with IC50 of 75 nM, Kd of <20 nM.
PC-42220

AZD5153 6-Hydroxy-2-naphthoic acid

BRD4 bromodomain inhibitor

AZD5153 is a potent, selective, bivalent and orally available BET/BRD4 bromodomain with IC50 of 5 nM.
PC-45507

PFI-4

BRPF1 inhibitor

PFI-4 is a potent, selective inhibitor of the BRPF1 bromodomain with pIC50 of 7.3.
PC-42109

BI-7273

BRD9 inhibitor

BI-7273 is a potent, selective and cell-permeable BRD9 bromodomain inhibitor with IC50 of 19 nM in Alpha assay.
PC-45780

PF-CBP1 hydrochloride

CBP/p300 inhibitor

PF-CBP1 hydrochloride is a potent, highly selective inhibitor of the CBP and p300 bromodomains with IC50 of 125 nM and 363 nM, respectively.

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