Ischemin |CAS:1357059-00-7 Probechem Biochemicals

Chemical Structure : Ischemin

Ischemin (CBP bromodomain inhibitor)

Catalog No.: PC-60199Not For Human Use, Lab Use Only.

Ischemin is a cell permeable CBP bromodomain inhibitor with Kd of 19 uM.

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Biological Activity

Ischemin is a cell permeable CBP bromodomain inhibitor with Kd of 19 uM.
Ischemin inhibits the acetyl-lysine binding activity of CBP, inhibits p53 interaction with CBP and decreases p53 transcriptional activity.
Ischemin protects against doxorubicin-induced apoptosis in cardiomyocytes in vitro.

Physicochemical Properties

M.Wt	335.378
Formula	C15H17N3O4S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	5-[(1E)-2-(2-Amino-4-hydroxy-5-methylphenyl)diazenyl]-2,4-dimethylbenzenesulfonic acid

References

1. Borah JC, et al. Chem Biol. 2011 Apr 22;18(4):531-41.

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Ischemin (CBP bromodomain inhibitor)

Biological Activity

Physicochemical Properties

References

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