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Cat. No. Product Name Information
PC-60932

BETi-211

BETi-211 is a novel potent small-molecule BET bromodomain (BRD) inhibitor that binds to BET proteins with Ki values of <1 nM.
PC-60930

Dual BET-Kinase inhibitor 3

BET inhibitor

Dual BET-Kinase inhibitor 3 is a potent, dual BET bromodomain-kinase inhibitor with IC50 of 34, 1.1 and 1.1 nM for BRD4 BD1, JAK2 and FLT-3, respectively.
PC-60857

CPI644

CREBBP/EP300

CPI644 (CPI-644) is a potent, selective, cell-active CREBBP/EP300 bromodomain inhibitor with IC50 of 0.18 uM for CREBBP.
PC-60856

CPI703

CBP/EP300 inhibitor

CPI-703 (CPI703) potent, selective, cell-active CBP/EP300 bromodomain inhibitor with IC50 of 0.47 uM for CBP.
PC-70222

GS-626510

GS-626510 (GS-6510, GS 6510, GS 626510) is a novel BET family bromodomains inhibitor with Kd of 0.5-2.8 nM for BRD2/3/4, and BRDT.
PC-60389

UMB-32

BRD4 inhibitor

UMB-32 is a potent, selective inhibitor of BRD4 with Kd of 550 nM, cellular IC50 of 724 nM.
PC-60388

UMB-136

UMB-136 (UMB136) is a novel bromodomain BRD4 inhibitor that significantly induces HIV-1 reactivation.
PC-60307

GNE-207

CBP/p300 inhibitor

GNE-207 (GNE207) is a novel potent, selective, orally active CBP/p300 bromodomain with IC50 of 1.0 nM.
PC-60306

GNE-781

CBP/p300 inhibitor

GNE-781 (GNE781) is a potent, selective, non-CNS penetrant, orally active CBP/p300 bromodomain inhibitor with IC50 of 0.94/1.2 nM in TR-FRET assays.
PC-60305

GNE-272

CBP/EP300 inhibitor

GNE-272 (GNE272) potent and selective the bromodomains of CBP/EP300 inhibitor with IC50 of 0.02 and 0.03 uM for CBP and EP300, respectively.
PC-60199

Ischemin

CBP bromodomain inhibitor

Ischemin is a cell permeable CBP bromodomain inhibitor with Kd of 19 uM.
PC-60198

Ischemin sodium

CBP bromodomain inhibitor

Ischemin sodium is a cell permeable CBP bromodomain inhibitor with Kd of 19 uM.

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