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Chemical Structure : FT-001
Catalog No.: PC-61740Not For Human Use, Lab Use Only.
FT-001 is a novel potent, orally acitve inhibitor of BET bromodomain with IC50 of 0.1 uM for BRD4 BD1.
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FT-001 (FT001) is a novel potent, orally acitve inhibitor of BET bromodomain with IC50 of 0.1 uM for BRD4 BD1.
FT-001 inhibits the expression of MYC in the MV-4-11 cell line with IC50 of 0.46 uM, shows anti-proliferative activity with IC50 of 0.22 uM.
FT-001 displays complete tumor growth inhibition in mouse MV-4-11 xenograft model.
| M.Wt | 467.584 | |
| Formula | C25H29N3O4S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Millan DS, et al. ACS Med Chem Lett. 2017 Jul 14;8(8):847-852.
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