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AZD6280

Chemical Structure : AZD6280

CAS No.: 942436-93-3

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AZD6280 (AZD-6280)

Catalog No.: PC-62765Not For Human Use, Lab Use Only.

AZD6280 is a potent, α2/3 functionally selective, partial GABAA receptor modulator with pKi of 7.7.

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5 mg $478 In stock
10 mg $758 In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

AZD6280 is a potent, α2/3 functionally selective, partial GABAA receptor modulator with pKi of 7.7.
AZD6280 exerts neutral antagonism at the α1-subunit and partial efficacy at the α2,3-subunits over the α5-subunit.
AZD6280 shows potential for the treatment of anxiety disorders.

Physicochemical Properties

M.Wt 366.421
Formula C20H22N4O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

4-amino-8-(2,5-dimethoxyphenyl)-N-propyl-3-cinnolinecarboxamide

References

1. Jucaite A, et al. Psychopharmacology (Berl). 2017 Feb;234(4):707-716.

2. Chen X, et al. J Clin Psychopharmacol. 2015 Feb;35(1):22-33.

3. Te Beek ET, et al. Clin Pharmacol Drug Dev. 2015 Mar;4(2):149-54.

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