Chemical Structure : Almorexant
CAS No.:
871224-64-5
Almorexant
(ACT-078573, ACT078573)
Catalog No. : PC-42704Not For Human Use, Lab Use Only.
Almorexant (ACT-078573) is a potent, dual Orexin receptor OX1/OX2 antagonist with Ki of 1.3/0.17 nM for hOX1/hOX2 respectively.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4270401
Biological Activity
Almorexant (ACT-078573) is a potent, dual Orexin receptor OX1/OX2 antagonist with Ki of 1.3/0.17 nM for hOX1/hOX2 respectively.
Physicochemical Properties
M.Wt
512.5632
Formula
C29H31F3N2O3
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
2(1H)-Isoquinolineacetamide, 3,4-dihydro-6,7-dimethoxy-N-methyl-α-phenyl-1-[2-[4-(trifluoromethyl)phenyl]ethyl]-, (αR,1S)-
References
1. Malherbe P, et al. Mol Pharmacol. 2009 Sep;76(3):618-31.
2. Malherbe P, et al. Mol Pharmacol. 2010 Jul;78(1):81-93.
3. Li A, et al. J Physiol. 2010 Aug 1;588(Pt 15):2935-44.
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