Artefenomel |CAS:1029939-86-3 Probechem Biochemicals

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Chemical Structure : Artefenomel

Artefenomel (OZ439)

Catalog No.: PC-62987Not For Human Use, Lab Use Only.

Artefenomel (OZ439) is a novel, next-generation antimalarial ozonide that demonstrates high potentcy against P. falciparum in vitro and P. berghei in vivo (K1/NF54, IC50=2.0/3.2 nM)..

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

Artefenomel (OZ439) is a novel, next-generation antimalarial ozonide that demonstrates high potentcy against P. falciparum in vitro and P. berghei in vivo (K1/NF54, IC50=2.0/3.2 nM).

Parasite Infection

Phase 2 Clinical

Physicochemical Properties

M.Wt	469.622
Formula	C28H39NO5
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	4-[2-(4-cis-Dispiro[cyclohexane-1,3'-[1,2,4]trioxolane-5',2''-tricyclo[3.3.1.13,7]decan]-4-ylphenoxy)ethyl]morpholine

References

1. Dong Y, et al. J Med Chem. 2017 Apr 13;60(7):2654-2668.

2. Kim HS, et al. J Med Chem. 2017 Apr 13;60(7):2651-2653.

3. Macintyre F, et al. BMC Med. 2017 Oct 9;15(1):181.

4. Yang T, et al. Antimicrob Agents Chemother. 2016 Jul 22;60(8):4501-10.

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Artefenomel (OZ439)

Biological Activity

Physicochemical Properties

References

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