BAZ2-ICR |CAS:1665195-94-7 Probechem Biochemicals

Chemical Structure : BAZ2-ICR

CAS No.: 1665195-94-7

BAZ2-ICR (BAZ2 ICR)

Catalog No.: PC-62269Not For Human Use, Lab Use Only.

BAZ2-ICR is a potent, selective and cell-active inhibitor of BAZ2A (Kd=109 nM, IC50=130 nM) and BAZ2B (Kd=170 nM, IC50=180 nM) bromodomains.

Packing	Price	Stock
10 mg	$128	In stock
25 mg	$198	In stock
50 mg	$328	In stock
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Biological Activity

BAZ2-ICR is a potent, selective and cell-active inhibitor of BAZ2A (Kd=109 nM, IC50=130 nM) and BAZ2B (Kd=170 nM, IC50=180 nM) bromodomains.
BAZ2-ICR demonstrates 15-fold selectivity for binding BAZ2A/B over CECR2 and >100-fold selectivity over all other bromodomains.

Physicochemical Properties

M.Wt	357.421
Formula	C20H19N7
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	4-[4-(1-methyl-1H-pyrazol-4-yl)-1-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-5-yl]-benzonitrile

References

1. Drouin L, et al. J Med Chem. 2015 Mar 12;58(5):2553-9.

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BAZ2-ICR (BAZ2 ICR)

Biological Activity

Physicochemical Properties

References

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