Catalog No.: PC-45764Not For Human Use, Lab Use Only.
BCTC is a highly potent, selective, CNS-penetrant TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 with IC50 values of 35 and 6 nM, respectively.
BCTC is a highly potent, selective, CNS-penetrant TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 with IC50 values of 35 and 6 nM, respectively.
BCTC shows selectivity against 63 other receptor, enzyme, transporter, and ion channel targets; orally bioavailable.
