BI-0252 |Cas:1818291-27-8 Buy BI-0252 from ProbeChem, Global Biochemicals Supplier

Chemical Structure : BI-0252

BI-0252 (BI 0252;BI0252)

Catalog No.: PC-60301Not For Human Use, Lab Use Only.

BI-0252 is a potent, highly selective, orally active MDM2-p53 interaction inhibitor with IC50 of 4 nM.

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Biological Activity

BI-0252 is a potent, highly selective, orally active MDM2-p53 interaction inhibitor with IC50 of 4 nM.
BI-0252 shows in vivo efficacy in a SJSA-1 xenograft model.

Physicochemical Properties

M.Wt	566.45
Formula	C30H26Cl2FN3O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	4-[(3S,3'S,3'aS,5'R,6'aS)-6-chloro-3'-(3-chloro-2-fluorophenyl)-1'-(cyclopropylmethyl)-2-oxo-1,2,3',3'a,4',5',6',6'a-octahydro-1'H-spiro[indole-3,2'-pyrrolo[3,2-b]pyrrole]-5'-yl]benzoic acid

References

1. Gollner A, et al. J Med Chem. 2016 Nov 23;59(22):10147-10162.

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BI-0252 (BI 0252;BI0252)

Biological Activity

Physicochemical Properties

References

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