BJG-05-039

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Chemical Structure : BJG-05-039

Catalog No.: PC-49535Not For Human Use, Lab Use Only.

BJG-05-039 is a PAK1-selective degrader consisting of NVS-PAK1-1 conjugated to lenalidomide, a recruiter of the E3 ubiquitin ligase substrate adaptor Cereblon.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

BJG-05-039 is a PAK1-selective degrader consisting of NVS-PAK1-1 conjugated to lenalidomide, a recruiter of the E3 ubiquitin ligase substrate adaptor Cereblon.

Physicochemical Properties

M.Wt	807.272
Formula	C40H42ClF3N8O5
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(3R)-3-((2-chloro-5-(2,2-difluoroethyl)-8-fluoro-5H-dibenzo[b,e][1,4]diazepin-11-yl)amino)-N-(7-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)heptyl)pyrrolidine-1-carboxamide

References

1. Hoi-Yee Chow, et al. J Med Chem. 2022 Nov 23. doi: 10.1021/acs.jmedchem.2c00756.

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BJG-05-039

Biological Activity

Physicochemical Properties

References

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