BJP-07-017-3

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Chemical Structure : BJP-07-017-3

Catalog No.: PC-23441Not For Human Use, Lab Use Only.

BJP-07-017-3 is a potent, selective, covalent, cell-permeable peptide Pin1 inhibitor (Ki=15 nM), IC50 of 9 nM in DELFIA assays, covalently targets Cys113, a highly conserved cysteine located in the Pin1 active site.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

Physicochemical Properties

M.Wt	709.25
Formula	C35H45ClN8O6
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-N-((S)-1-(((S)-1-amino-1-oxo-5-ureidopentan-2-yl)amino)-3-(1H-indol-3-yl)-1-oxopropan-2-yl)-1-(N-(2-chloroacetyl)-N-methyl-L-phenylalanyl)piperidine-2-carboxamide

References

1. B. J. Pinch et al., Identification of a potent and selective covalent Pin1 inhibitor. Nat. Chem. Biol. 16, 979–987 (2020).

2. Alboreggia G, et al. Proc Natl Acad Sci U S A. 2024 Nov 19;121(47):e2403330121.

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BJP-07-017-3

Biological Activity

Physicochemical Properties

References

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