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BL-6020 979

Chemical Structure : BL-6020 979

CAS No.:

BL-6020 979 (SNT207979;BL-6020/979)

Catalog No.: PC-61572Not For Human Use, Lab Use Only.

BL-6020/979 (SNT207979) is an orally available, selective, potent MC4R antagonist with IC50 of 19 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    BL-6020/979 (SNT207979) is an orally available, selective, potent MC4R antagonist with IC50 of 19 nM.
    BL-6020/979 (SNT207979) weakly binds to MC-3 and MC-5 receptors with IC50 of 2.7 uM and 0.89 uM, respectively, >10,000-fold selectivity over MC-1R;.
    BL-6020/979 (SNT207979) demonstrates in animal models and presents a promising candidate suitable for further development towards a first-in-class treatment option for cachexia.

    Physicochemical Properties

    M.Wt
    Formula
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    References

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