Welcome to ProbeChem!Global Supplier of Chemical Probes, Inhibitors & Agonists.
Chemical Structure : BP 897
CAS No.: 314776-92-6
Catalog No.: PC-61736Not For Human Use, Lab Use Only.
BP 897 is the first, potent, selective partial dopamine D3 receptor agonist with Ki of 0.92 nM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $128 | In stock | |
| 25 mg | $218 | In stock | |
| 50 mg | $368 | In stock | |
| 100 mg | Get quote |
Bulk size, bulk discount!
E-mail: sales@probechem.com
Tech Support: tech@probechem.com
BP 897 is the first, potent, selective partial dopamine D3 receptor agonist with Ki of 0.92 nM.
BP 897 displays 70 times lower affinity for D2 (Ki=61 nM), low affinities for D1 and D4 (Ki= 3 and 0.3 uM) and α1 and α2 adrenergic receptor (Ki=60 and 83 nM), negligible affinities (Ki>1 uM) for muscarinic, histamine and opiate receptors.
BP 897 inhibits cocaine-seeking behaviour that depends upon the presentation of drug-associated cues, without having any intrinsic, primary rewarding effects.
| M.Wt | 417.553 | |
| Formula | C26H31N3O2 | |
| Appearance | Solid | |
| Storage |
|
|
| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2-naphthamide |
|
1. Pilla M, et al. Nature. 1999 Jul 22;400(6742):371-5.
2. Wood MD, et al. Eur J Pharmacol. 2000 Oct 27;407(1-2):47-51.
3. Wicke K, et al. Eur J Pharmacol. 2001 Jul 20;424(2):85-90.
Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright
