BPTF inhibitor BZ1

Chemical Structure : BPTF inhibitor BZ1

Catalog No.: PC-72758Not For Human Use, Lab Use Only.

BPTF inhibitor BZ1 is a potent, selective, cell-active inhibitor of bromodomain PHD finger transcription factor (BPTF) with Kd of 6.3 nM, >350-fold selectivity over BET bromodomains.

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Biological Activity

BPTF inhibitor BZ1 is a potent, selective, cell-active inhibitor of bromodomain PHD finger transcription factor (BPTF) with Kd of 6.3 nM, >350-fold selectivity over BET bromodomains.
BPTF inhibitor BZ1 sensitizes 4T1 breast cancer cells to doxorubicin but not BPTF knockdown cells, suggesting a specificity to BPTF.

Physicochemical Properties

M.Wt	278.74
Formula	C13H15ClN4O
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Month
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Chemical Name/SMILES

References

1. Huda Zahid, et al. J Med Chem. 2021 Sep 23;64(18):13902-13917.

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