BR103 | C3aR inhibitor | Probechem Biochemicals

Chemical Structure : BR103

BR103 (BR 103)

Catalog No.: PC-61771Not For Human Use, Lab Use Only.

BR103 is a potent, metabolically stable and highly selective small molecule agonist of complement C3a receptor (C3aR) with EC50 of 22 nM.

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Biological Activity

BR103 is a potent, metabolically stable and highly selective small molecule agonist of complement C3a receptor (C3aR) with EC50 of 22 nM.
BR103 displays high selectivity for C3aR over C5aR.
BR103 induces paw oedema and mast cell activation in vivo in rats.

Physicochemical Properties

M.Wt	448.527
Formula	C24H28N6O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(2-benzhydryl-5-methyl-1H-imidazole-4-carbonyl)-L-arginine

References

1. Lohman RJ, et al. Nat Commun. 2017 Aug 24;8(1):351.

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BR103 (BR 103)

Biological Activity

Physicochemical Properties

References

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