BRD-IN-26 |CAS:1915012-19-9 Probechem Biochemicals

Chemical Structure : BRD-IN-26

BRD-IN-26 (PB1(5) inhibitor)

Catalog No.: PC-62277Not For Human Use, Lab Use Only.

BRD-IN-26 is a potent bromodomain inhibitor that binds the fifth bromodomain of PB1 (PB1(5)) with a KD of 124 nM, SMARCA2B and SMARCA4 with KD values of 262 and 417 nM, respectively.

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Biological Activity

BRD-IN-26 is a potent bromodomain inhibitor that binds the fifth bromodomain of PB1 (PB1(5)) with a KD of 124 nM, SMARCA2B and SMARCA4 with KD values of 262 and 417 nM, respectively.
BRD-IN-26 displays excellent selectivity over other bromodomains.

Physicochemical Properties

M.Wt	330.816
Formula	C17H19ClN4O
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(E)-6-chloro-3-((4-methylpiperazin-1-yl)methylene)-2,3-dihydropyrrolo[1,2-a]quinazolin-5(1H)-one

References

1. Sutherell CL, et al. J Med Chem. 2016 May 26;59(10):5095-101.

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BRD-IN-26 (PB1(5) inhibitor)

Biological Activity

Physicochemical Properties

References

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