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Chemical Structure : BRD4 D1 inhibitor 30
Catalog No.: PC-72261Not For Human Use, Lab Use Only.
BRD4 D1 inhibitor 30 is a high-affinity, BRD4 D1-selective chemical probe with Kd of 18 nM, 500-fold selectivity against BRD2 D1 and BRD4 D2.
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BRD4 D1 inhibitor 30 is a high-affinity, BRD4 D1-selective chemical probe with Kd of 18 nM, 500-fold selectivity against BRD2 D1 and BRD4 D2.
BRD4 D1 inhibitor 30 down regulated inflammation, IL-8 and chemokine in cell based assays, but was unable to reduce c-Myc expression at low concentration in multiple myeloma cells.
| M.Wt | 578.684 | |
| Formula | C32H37F3N6O | |
| Appearance | Solid | |
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1. Huarui Cui, et al. J Med Chem. 2022 Feb 10;65(3):2342-2360.
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