BRD9-IN-28 |CAS:1947372-67-9 Probechem Biochemicals

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Chemical Structure : BRD9-IN-28

BRD9-IN-28

Catalog No.: PC-62938Not For Human Use, Lab Use Only.

BRD9-IN-28 is a highly potent and selective BRD7/9 bromodomain inhibitor with pIC50 of 6.9, Kd of 68 nM for BRD9.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

BRD9-IN-28 is a highly potent and selective BRD7/9 bromodomain inhibitor with pIC50 of 6.9, Kd of 68 nM for BRD9.
BRD9-IN-28 is slightly less potent against BRD7 (Kd=368 nM) and completely inactive against BAZ2B, little affinity across BRD proteins from sub-families 1-3 and 5-8, including BAZ2A and BAZ2B.
BRD9-IN-28 shows weak affinity for the BRDs from CBP, p300 and FALZ.

Physicochemical Properties

M.Wt	360.417
Formula	C21H20N4O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	1-(1-(imidazo[1,2-a]pyridin-5-yl)-7-morpholinoindolizin-3-yl)ethan-1-one

References

1. Duncan. A. Hay, et al. Med. Chem. Commun., 2015, DOI: 10.1039/C5MD00152H.

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BRD9-IN-28

Biological Activity

Physicochemical Properties

References

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