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Chemical Structure : BRD9539
CAS No.: 1374601-41-8
Catalog No.: PC-49729Not For Human Use, Lab Use Only.
BRD9539 is a small molecule inhibitor of histone hethyltransferase of G9a (euchromatin histone methyltransferase 2, EHMT2) with IC50 of 6.3 uM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $98 | In stock | |
| 25 mg | $158 | In stock | |
| 50 mg | $258 | In stock | |
| 100 mg | Get quote |
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BRD9539 is a small molecule inhibitor of histone hethyltransferase of G9a (euchromatin histone methyltransferase 2, EHMT2) with IC50 of 6.3 uM.
BRD9539 also inhibits PRC2 activity with a similar IC50, displays no inhibition aginst SUV39H1 and DNMT1.
BRD9539 is a more potent biochemical inhibitor than its methyl-ester analogue BRD4770.
| M.Wt | 399.45 | |
| Formula | C24H21N3O3 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
2-benzamido-1-(3-phenylpropyl)-1H-benzo[d]imidazole-5-carboxylic acid |
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1. Yuan Yuan, et al. ACS Chem Biol. 2012 Jul 20;7(7):1152-7.
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