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BRD9539

Chemical Structure : BRD9539

CAS No.: 1374601-41-8

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BRD9539 (BRD 9539)

Catalog No.: PC-49729Not For Human Use, Lab Use Only.

BRD9539 is a small molecule inhibitor of histone hethyltransferase of G9a (euchromatin histone methyltransferase 2, EHMT2) with IC50 of 6.3 uM.

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Biological Activity

BRD9539 is a small molecule inhibitor of histone hethyltransferase of G9a (euchromatin histone methyltransferase 2, EHMT2) with IC50 of 6.3 uM.
BRD9539 also inhibits PRC2 activity with a similar IC50, displays no inhibition aginst SUV39H1 and DNMT1.
BRD9539 is a more potent biochemical inhibitor than its methyl-ester analogue BRD4770.

Physicochemical Properties

M.Wt 399.45
Formula C24H21N3O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2-benzamido-1-(3-phenylpropyl)-1H-benzo[d]imidazole-5-carboxylic acid

References

1. Yuan Yuan, et al. ACS Chem Biol. 2012 Jul 20;7(7):1152-7.

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