BRPF1B TRIM24-IN-34 |CAS:1242907-48-7 Probechem Biochemicals

Chemical Structure : BRPF1B TRIM24-IN-34

BRPF1B TRIM24-IN-34

Catalog No.: PC-62285Not For Human Use, Lab Use Only.

BRPF1B TRIM24-IN-34 is a selective BRPF1B/TRIM24 dual inhibitor that binds with KD of 137 and 222 nM, respectively.

Packing	Price	Stock	Quantity
25 mg		Get quote
100 mg		Get quote
200 mg		Get quote
1 g		Get quote

Get Quotation Now

* Please select Quantity before adding items.

or Bulk Inquiry

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Biological Activity

BRPF1B TRIM24-IN-34 is a selective BRPF1B/TRIM24 dual inhibitor that binds with KD of 137 and 222 nM, respectively.
BRPF1B TRIM24-IN-34 exhibits good selectivity over other bromodomains.
BRPF1B TRIM24-IN-34 showes no significant cytotoxicity in a panel of cancer cell lines (GI50>10 uM).

Physicochemical Properties

M.Wt	499.538
Formula	C24H25N3O7S
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3,4-dimethoxy-N-(6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)benzenesulfonamide

References

1. Bennett J, et al. J Med Chem. 2016 Feb 25;59(4):1642-7.

Overnight Delivery
Fast & Safe Delivery Worldwide
Rewards Program

About Us

Our Services

Site Map

Join with Us
Product Use Citations

Pharmacological Glossary Abbreviations

Abbreviations

Quality Manual

Inquiry Form
How to Order

Terms & Conditions

Credit Card Payment

Shipping Rates & Policies

Privacy Policy
sales@probechem.com