BRS-3 agonist Compound A racemate

Chemical Structure : BRS-3 agonist Compound A racemate

Catalog No.: PC-61218Not For Human Use, Lab Use Only.

A potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist with EC50 of 270/130 nM for human/rat BRS-3, respectively.

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Biological Activity

A potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist with EC50 of 270/130 nM for human/rat BRS-3, respectively; displays no activity against GRPR (BRS-1) and NMBR (BRS-2) (EC50>10 uM).

Physicochemical Properties

M.Wt	428.532
Formula	C27H28N2O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	6-benzyl-N-tert-butyl-9-methoxy-7-oxo-6,7-dihydro-5H-dibenzo[c,e]azepine-5-carboxamide

References

1. Nio Y, et al. Endocrinology. 2017 May 1;158(5):1298-1313.

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