| Cat. No. |
Product Name |
Information |
| PC-20957 |
DSO-5a
BRS-3 agonist
|
DSO-5a (Dimethyl shikonin oxime 5a) is a potent, selective agonist pf bombesin receptor subtype-3 (BB3, BRS-3) with pEC50 of 8.4 (IP-1 accumulation in hBB3-H1299 cells). |
| PC-38792 |
MK-5046
BRS-3 agonist
|
MK-5046 a potent, selective small molecule agonist of BRS-3 (bombesin receptor subtype-3) with Ki and EC50 values of 3.7 and 14 nM (hBRS-3), respectively. |
| PC-61219 |
RC-3095
GRPR (BRS-1) inhibitor
|
RC-3095 is a potent, peptide bombesin/gastrin releasing peptide (GRPR,BRS-1) antagonist. |
| PC-61216 |
BRS-3 agonist Compound A
BRS-3 agonist
|
BRS-3 agonist Compound A (Compound-A) is a potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist with EC50 of 250/100 nM for human/rat BRS-3, respectively. |
| PC-61215 |
Bantag-1 trifluoroacetate
BRS-3 antagonist
|
Bantag-1 trifluoroacetate is a potent, highly selective, peptide bombesin receptor subtype-3 (BRS-3) antagonist with IC50 of 2-8 nM for human and rodent BRS-3. |
| PC-24417 |
Aurantiamide
GRPR antagonist
|
Aurantiamide is a potent, non-covalent, orally active, BBB-permeable antagonist of gastrin-releasing peptide receptor (GRPR), shows anti-inflammatory and neuroprotective effects. |
| PC-21220 |
PD168368
NMB-R antagonist
|
PD168368 is a potent, competitive, and selective neuromedin B receptor (NMB-R) antagonist with Ki of 15 nM, IC50 of 96 nM. |
| PC-61218 |
BRS-3 agonist Compound A racemate
|
A potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist with EC50 of 270/130 nM for human/rat BRS-3, respectively. |
| PC-61217 |
(S)-BRS-3 agonist Compound A
|
The distomer of BRS-3 agonist Compound A, shows no activity for bombesin receptor subtype-3 (BRS-3) with EC50>10 uM.. |
