| Cat. No. |
Product Name |
CAS No. |
Information |
| PC-61219 |
RC-3095
|
138147-78-1 |
A potent, peptide bombesin/gastrin releasing peptide (GRPR,BRS-1) antagonist.. |
| PC-61218 |
BRS-3 agonist Compound A racemate
|
|
A potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist with EC50 of 270/130 nM for human/rat BRS-3, respectively. |
| PC-61217 |
(S)-BRS-3 agonist Compound A
|
|
The distomer of BRS-3 agonist Compound A, shows no activity for bombesin receptor subtype-3 (BRS-3) with EC50>10 uM.. |
| PC-61216 |
BRS-3 agonist Compound A
|
|
A potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist with EC50 of 250/100 nM for human/rat BRS-3, resp+H1437+M1438. |
| PC-61215 |
Bantag-1 trifluoroacetate
|
|
A potent, highly selective, peptide bombesin receptor subtype-3 (BRS-3) antagonist with IC50 of 2-8 nM for human and rodent BRS-3, displays 1000-fold selectivity over hNMBR and hGRPR, increases food intake and produces an obesity phenotype in mice.. |
